Contextualising Trifecta ADC Design & Advancing Next-Generation Branched Linker ADC Development

  • Applying a trifecta approach to design a fit-for-purpose linker for haematologic ADCs, with preclinical insights from Debio-1562M incorporating MLINKSELECT DM1
  • Developing and implementing branched linker technology for next-generation dual payload ADCs in solid tumours
  • Recapping lessons learned in advancing high-DAR ADCs from discovery to the clinic